Synthesis and applications of β-aminoethanesulfonyl azides

Arwin J. Brouwer; Remco Merkx; Katarzyna Dabrowska; Dirk T.S. Rijkers; Rob M.J. Liskamp

doi:10.1055/s-2006-926273

Synthesis and applications of β-aminoethanesulfonyl azides

Arwin J. Brouwer
, Remco Merkx
, Katarzyna Dabrowska
, Dirk T.S. Rijkers
, Rob M.J. Liskamp^*

^*Corresponding author for this work

Chemical Biology and Drug Discovery

Utrecht University

Research output: Contribution to journal › Article › Academic › peer-review

Abstract

A very efficient method for the synthesis of β-aminoethanesulfonyl azides is descibed. These aliphatic sulfonyl azides are accessible starting from a variety of protected amino acids, including those having functionalized side chains. Furthermore, these sulfonyl azides can be coupled to thio acids, and can be substituted with different aliphatic amines.

Original language	English
Pages (from-to)	455-460
Number of pages	6
Journal	Synthesis
Issue number	3
DOIs	https://doi.org/10.1055/s-2006-926273
Publication status	Published - 1 Feb 2006

Keywords

Amino acid
Sulfonamides
Sulfonyl azide
Sulfonyl chloride

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10.1055/s-2006-926273

Cite this

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title = "Synthesis and applications of β-aminoethanesulfonyl azides",

abstract = "A very efficient method for the synthesis of β-aminoethanesulfonyl azides is descibed. These aliphatic sulfonyl azides are accessible starting from a variety of protected amino acids, including those having functionalized side chains. Furthermore, these sulfonyl azides can be coupled to thio acids, and can be substituted with different aliphatic amines.",

keywords = "Amino acid, Sulfonamides, Sulfonyl azide, Sulfonyl chloride",

author = "Brouwer, \{Arwin J.\} and Remco Merkx and Katarzyna Dabrowska and Rijkers, \{Dirk T.S.\} and Liskamp, \{Rob M.J.\}",

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AU - Brouwer, Arwin J.

AU - Merkx, Remco

AU - Dabrowska, Katarzyna

AU - Rijkers, Dirk T.S.

AU - Liskamp, Rob M.J.

PY - 2006/2/1

Y1 - 2006/2/1

N2 - A very efficient method for the synthesis of β-aminoethanesulfonyl azides is descibed. These aliphatic sulfonyl azides are accessible starting from a variety of protected amino acids, including those having functionalized side chains. Furthermore, these sulfonyl azides can be coupled to thio acids, and can be substituted with different aliphatic amines.

AB - A very efficient method for the synthesis of β-aminoethanesulfonyl azides is descibed. These aliphatic sulfonyl azides are accessible starting from a variety of protected amino acids, including those having functionalized side chains. Furthermore, these sulfonyl azides can be coupled to thio acids, and can be substituted with different aliphatic amines.

KW - Amino acid

KW - Sulfonamides

KW - Sulfonyl azide

KW - Sulfonyl chloride

UR - https://www.scopus.com/pages/publications/32644454133

U2 - 10.1055/s-2006-926273

DO - 10.1055/s-2006-926273

M3 - Article

AN - SCOPUS:32644454133

SN - 0039-7881

SP - 455

EP - 460

JO - Synthesis

JF - Synthesis

IS - 3

ER -

Synthesis and applications of β-aminoethanesulfonyl azides

Abstract

Keywords

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