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Insights into PPARγ phosphorylation and its inhibition mechanism
Roberta Montanari
, Davide Capelli
, Keiko Yamamoto
, Hirono Awaishima
, Kimina Nishikata
,
Arjan Barendregt
,
Albert J R Heck
, Fulvio Loiodice
, Fabio Altieri
, Alessandro Paiardini
, Alessandro Grotessi
, Luciano Pirone
, Emilia Maria Pedone
, Franck Peiretti
, Jean Michel Brunel
, Toshimasa Itoh
, Giorgio Pochetti
Biomolecular Mass Spectrometry and Proteomics
Sub Biomolecular Mass Spectrometry and Proteomics
Biomolecular Mass Spectrometry and Proteomics
Biomolecular Mass Spectrometry and Proteomics
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Keyphrases
Phosphorylation
100%
Inhibition Mechanism
100%
Antidiabetic Drugs
66%
Cyclin-dependent Kinase 5 (Cdk5)
66%
X-ray
33%
Conformational Change
33%
Protein-protein Docking
33%
Type 2 Diabetes Prevention
33%
Molecular Dynamics Simulation
33%
Phosphorylation Sites
33%
Agonism
33%
Metabolic Syndrome
33%
Site-directed mutagenesis
33%
Multidisciplinary Approach
33%
Nuclear Receptor
33%
Undesirable Side Effects
33%
Diabetes Syndrome
33%
Immunology and Microbiology
Conformational Transition
100%
Site Directed Mutagenesis
100%
X Ray
100%
Pharmacology, Toxicology and Pharmaceutical Science
Peroxisome Proliferator Activated Receptor
100%
Antidiabetic Agent
25%
Site-Directed Mutagenesis
12%
Side Effect
12%
Docking Protein
12%
Cell Nucleus Receptor
12%
Metabolic Syndrome X
12%
Non Insulin Dependent Diabetes Mellitus
12%
Biochemistry, Genetics and Molecular Biology
Peroxisome Proliferator-Activated Receptor
100%
X Ray
12%
Conformational Change
12%
Site-Directed Mutagenesis
12%
Signal Recognition Particle Receptor
12%
Nuclear Receptor
12%